TABLE 1

Sulfonylurea receptor (SUR)1 and SUR2 activators and inhibitors

SUR1 and SUR2 activatorsSUR1 and SUR2 inhibitors
PinacidilTolbutamide
Nicorandil#Glibenclamide
DiazoxideAcetohexamide
CromakalimTolazamide
Minoxidil#Glipizide
Chlorpropamide
Glyburide

Information from DrugBank [17] and the International Union of Basic and Clinical Pharmacology [18]. #: SUR activators with additional vasodilator properties were identified.